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Innovative Medicines & Omics                                           SARS-CoV-2 inhibition by quinolines



               Chem. 2023;15(17):1569-1582.                       doi: 10.3390/ph15010021

               doi: 10.4155/fmc-2023-0169                      35.  Laboratory Biosafety Guidance Related to Coronavirus
                                                                  Disease  (COVID-19):  Interim  Guidance;  2021.  Available
            25.  Vausselin T, Séron K, Lavie M, et al. Identification of a new   from: https://www.who.int/publications/i/item/who-wpe-
               benzimidazole derivative as an antiviral against hepatitis C
               virus. J Virol. 2016;90(19):8422-8434.             gih-2021.1 [Last accessed on 2023 Sep 10].
                                                                                            pro
                                                               36.  Jin Z, Du X, Xu Y, et al. Structure of M  from SARS-CoV-2 and
               doi: 10.1128/JVI.00404-16
                                                                  discovery of its inhibitors. Nature. 2020;582(7811):289-293.
            26.  Ekins S, Freundlich JS, Clark AM, Anantpadma M, Davey  RA,
               Madrid P. Machine learning models identify molecules active      doi: 10.1038/s41586-020-2223-y
               against the Ebola virus in vitro. F1000Res. 2015;4:1091.  37.  Goyal B, Goyal D. Targeting the dimerization of the main
                                                                  protease of coronaviruses: A  potential broad-spectrum
               doi: 10.12688/f1000research.7217.3
                                                                  therapeutic strategy. ACS Comb Sci. 2020;22(6):297-305.
            27.  Hu Q, Xiong Y, Zhu GH,  et al. The SARS-CoV-2 main      doi: 10.1021/acscombsci.0c00058
               protease (Mpro): Structure, function, and emerging
               therapies for COVID-19. MedComm (2020). 2022;3(3):e151.  38.  Uzunova K, Filipova E, Pavlova V,  et al. Insights into
                                                                  antiviral mechanisms of remdesivir, lopinavir/ritonavir and
               doi: 10.1002/mco2.151
                                                                  chloroquine/hydroxychloroquine affecting the  new SARS-
            28.  Zhang L, Lin D, Sun X,  et al. Crystal structure of SARS-  CoV-2. Biomed Pharmacother. 2020;131:110668.
               CoV-2 main protease provides a basis for design of improved
               a-ketoamide inhibitors. Science. 2020;368(6489):409-412.     doi: 10.1016/j.biopha.2020.110668
                                                               39.  Patel TK, Patel PB, Barvaliya M, et al. Efficacy and safety
               doi: 10.1126/science.abb3405
                                                                  of lopinavir-ritonavir in COVID-19: A  systematic review
            29.  Achutha AS, Pushpa VL, Suchitra S. Theoretical insights   of  randomized  controlled  trials.  J  Infect  Public  Health.
               into the anti-SARS-CoV-2 activity of chloroquine and its   2021;14(6):740-748.
               analogs and in silico screening of main protease inhibitors.      doi: 10.1016/j.jiph.2021.03.015
               J Proteome Res. 2020;9(11):4706-4717.
                                                               40.  Habler  K, Brügel M,  Teupser  D,  et al. Simultaneous
               doi: 10.1021/acs.jproteome.0c00683
                                                                  quantification of seven repurposed COVID-19 drugs
            30.  Carmo AM, Silva FM, Machado PA,  et al. Synthesis of   remdesivir (plus metabolite GS-441524), chloroquine,
               4-aminoquinoline analogues and their platinum(II)   hydroxychloroquine, lopinavir, ritonavir, favipiravir and
               complexes as new antileishmanial and antitubercular agents.   azithromycin by a two-dimensional isotope dilution
               Biomed Pharmacother. 2011;65(3):204-209.           LC-MS/MS method in human serum. J Pharm Biomed Anal.
                                                                  2021;196:113935.
               doi: 10.1016/j.biopha.2011.01.003
                                                                  doi: 10.1016/j.jpba.2021.113935
            31.  Calixto  SL,  Glanzmann  N,  Xavier  Silveira  MM,  et al.
               Novel organic salts based on quinoline derivatives: The   41.  Lipinski CA, Lombardo F, Dominy BW, et al. Experimental
               in vitro activity trigger apoptosis inhibiting autophagy in   and computational approaches to estimate solubility and
               Leishmania spp. Chem Biol Interact. 2018;293:141-151.  permeability in drug discovery and development settings.
                                                                  [The article was originally published in Adv Drug Deliv Rev.
               doi: 10.1016/j.cbi.2018.08.003
                                                                  1997;23:3-25]. Adv Drug Deliv Rev. 2001;46(1-3):3-26.
            32.  Dludla PV, Jack B, Viraragavan A, et al. A dose-dependent
               effect of dimethyl sulfoxide on lipid content, cell viability      doi: 10.1016/S0169-409X(00)00129-0
               and oxidative stress in 3T3-L1 adipocytes.  Toxicol   42.  Veber DF, Johnson SR, Cheng HY, Smith BR, Ward
               Rep. 2018;5:1014-1020.                             KW, Kopple KD. Molecular properties that influence
                                                                  the oral bioavailability of drug candidates.  J  Med Chem.
               doi: 10.1016/j.toxrep.2018.10.002
                                                                  2002;45(12):2615-2623.
            33.  Fintelman-Rodrigues N, Sacramento CQ, Ribeiro Lima C,
               et al. Atazanavir, alone or in combination with ritonavir,      doi: 10.1021/jm020017n
               inhibits SARS-CoV-2 replication and proinflammatory   43.  Kelder J, Grootenhuis PD, Bayada DM, Delbressine LP,
               cytokine production.  Antimicrob  Agents  Chemother.   Ploemen  JP.  Polar  molecular  surface  as  a  dominating
               2020;64(10):e00825-20.                             determinant for oral absorption and brain penetration of
               doi: 10.1128/AAC.00825-20                          drugs. Pharm Res. 1999;16(10):1514-1519.
                                                                  doi: 10.1023/A:1015040217741
            34.  Chaves OA, Sacramento CQ, Ferreira AC, et al. Atazanavir
               is a competitive inhibitor of SARS-CoV-2 M , impairing   44.  Zhu Y, Chidekel A, Shaffer TH. Cultured human airway
                                                 pro
               variants replication  in vitro  and  in vivo.  Pharmaceuticals   epithelial cells (Calu-3): A  model of human respiratory
               (Basel). 2021;15(1):21.                            function, structure, and inflammatory responses. Crit Care


            Volume 1 Issue 1 (2024)                        104                               doi: 10.36922/imo.3442
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